描述:2'- Fluoro-NTP在新药开发和研究中的利用数量逐渐增加。同时也用于寡核苷酸适配子和siRNA的设计和合成,增强外源DNA在生物体内的稳定性。
2'- Fluoro-NTP
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2'- Fluoro-NTP在新药开发和研究中的利用数量逐渐增加。zui近,2' Fluoro ATP被证实是研究制药适用激酶时筛选ATP需求酶的通用工具。2' Fluoro NTPs能与酶兼容提高DNA和RNA在体内的稳定性。2' Fluoro NTPs常用于寡核苷酸适配子和siRNA的设计和合成,因为它在体内的传送增加了靶分子的亲和力,阻碍核酸酶的作用,同时降低免疫反应。2' Fluoro NTP是非常不错的DNA和RNA聚合酶,包括广泛使用的T7 RNA聚合酶的底物。
2' Fluoro Nucleoside Triphosphates | |||
N-1007-1 | 2'-Fluoro-2'-deoxyadenosine-5'-TP | 1umole | 1317.5 |
N-1007-5 | 2'-Fluoro-2'-deoxyadenosine-5'-TP | 5umoles | 6205 |
N-1007-10 | 2'-Fluoro-2'-deoxyadenosine-5'-TP | 10umoles | 10625 |
N-1008-1 | 2'-Fluoro-2'-deoxycytidine-5'-TP | 1umole | 892.5 |
N-1008-5 | 2'-Fluoro-2'-deoxycytidine-5'-TP | 5umoles | 4335 |
N-1008-10 | 2'-Fluoro-2'-deoxycytidine-5'-TP | 10umoles | 7055 |
N-1009-1 | 2'-Fluoro-2'-deoxyguanosine-5'-TP | 1umole | 1657.5 |
N-1009-5 | 2'-Fluoro-2'-deoxyguanosine-5'-TP | 5umoles | 7905 |
N-1009-10 | 2'-Fluoro-2'-deoxyguanosine-5'-TP | 10umoles | 14450 |
N-1010-1 | 2'-Fluoro-2'-deoxyuridine-5'-TP | 1umole | 892.5 |
N-1010-5 | 2'-Fluoro-2'-deoxyuridine-5'-TP | 5umoles | 4335 |
N-1010-10 | 2'-Fluoro-2'-deoxyuridine-5'-TP | 10umoles | 7055 |
N-1055-1 | 2'-Fluoro-thymidine-5'-TP | 1umole | 1317.5 |
N-1055-5 | 2'-Fluoro-thymidine-5'-TP | 5umoles | 6205 |
N-1055-10 | 2'-Fluoro-thymidine-5'-TP | 10umoles | 10625 |